Sunday April 21, 2024 |
17:30 | Registration |
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19:30 | Dinner at the Hotel |
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21:00 | Get Together at the Castle Bar |
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Monday April 22, 2024 |
07:15 | Breakfast |
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08:15 | Opening Ceremony |
Prof. Laura HEITMAN (UNIVERSITY OF LEIDEN, Leiden, The Netherlands) |
08:30 | Physicochemical Property Considerations in Modern Drug Discovery and Implications for Hit Finding and Library Design - Part 1 |
Prof. Mike WARING (NEWCASTLE UNIVERSITY, Newcastle upon Tyne, United Kingdom) Dr Hannah STEWART (NEWCASTLE UNIVERSITY, Newcastle Upon Tyne, United Kingdom) |
10:00 | Coffee Break |
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10:30 | Physicochemical Property Considerations in Modern Drug Discovery and Implications for Hit Finding and Library Design - Part 2 |
Prof. Mike WARING (NEWCASTLE UNIVERSITY, Newcastle upon Tyne, United Kingdom) Dr Hannah STEWART (NEWCASTLE UNIVERSITY, Newcastle Upon Tyne, United Kingdom) |
12:00 | Lunch & Group Picture |
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13:30 | What Can We Learn from 20+ years of Fragment Based Drug Discovery and What Are the Future Opportunities? - Part 1 |
Dr Christopher JOHNSON (ASTEX PHARMACEUTICALS, Cambridge, United Kingdom) |
15:00 | Coffee Break |
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15:30 | What Can We Learn from 20+ years of Fragment Based Drug Discovery and What Are the Future Opportunities? - Part 2 |
Dr Christopher JOHNSON (ASTEX PHARMACEUTICALS, Cambridge, United Kingdom) |
17:00 | Day End |
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18:00 | Walking tour through Leiden |
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19:30 | Dinner in Leiden |
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Tuesday April 23, 2024 |
08:30 | Enabling Drug Discovery Projects with Encoded Library Technologies - Part 1 |
Dr Frederic BERST (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Basel, Switzerland) Dr Christoph DUMELIN (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Basel, Switzerland) |
10:00 | Coffee Break |
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10:30 | Enabling Drug Discovery Projects with Encoded Library Technologies - Part 2 |
Dr Frederic BERST (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Basel, Switzerland) Dr Christoph DUMELIN (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Basel, Switzerland) |
12:00 | Lunch |
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13:30 | Design of Multifunctional Conjugates for the Targeting of Non-coding RNAs: Anticancer and Antimicrobial Applications |
Dr Maria DUCA (UNIVERSITY OF CÔTE D'AZUR, Nice, France) |
15:00 | Coffee Break |
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15:30 | Activity Based Profiling as Tool in Medicinal Chemistry |
Prof. Mario VAN DER STELT (UNIVERSITY OF LEIDEN, Leiden, The Netherlands) |
17:00 | Day End |
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19:30 | Dinner at the hotel |
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21:00 | Get Together at the Castle Bar |
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Wednesday April 24, 2024 |
07:00 | Breakfast |
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08:30 | General Considerations for Covalent Drug Discovery Exemplified with Acalabrutinib |
Dr Gerjan DE BRUIN (ACERTA PHARMA, Oss, The Netherlands) |
10:00 | Coffee Break |
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10:30 | Discovery of Zosurabalpin |
Dr Patrizio MATTEI (ROCHE INNOVATION CENTER BASEL, Basel, Switzerland) |
12:00 | Wrap up and Lunch |
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